Répertoire du corps professoral
Vincenzo Di Marzo
Professeur titulaire
vincenzo.dimarzo@criucpq.ulaval.ca
Pavillon Ferdinand-Vandry
1050, avenue de la Médecine
Local 4211
Professeur titulaire
vincenzo.dimarzo@criucpq.ulaval.ca
Pavillon des Services
2440, boul Hochelaga
Local 1705
Institut sur la nutrition et les aliments fonctionnels (INAF)
Programme: Regroupements stratégiques NT
Organisme(s) subventionnaire(s): Institut national de recherche scientifique (INRS), Fonds de recherche du Québec - Nature et technologies, Université Laval - Fonds internes, Université McGill, Université du Québec à Rimouski, Université de Sherbrooke
Établissement tête: Université Laval
Du 1 avril 2017
au 31 mars 2024
FMÉD --- Support de Sentinelle Nord à l'Unité mixte internationale sur la recherche chimique et biomoléculaire de microbiome
Programme: Fonds d'excellence en recherche Apogée Canada
Organisme(s) subventionnaire(s): Secrétariat des programmes interorganismes à l’intention des établissements
Établissement tête: Université Laval
Du 1 juin 2017
au 31 août 2023
Canada Excellence Research Chair on the microbiome-endocannabinoidome connection in metabolic health
Programme: Programme de chaires d'excellence en recherche du Canada
Organisme(s) subventionnaire(s): Instituts de recherche en santé du Canada
Établissement tête: Université Laval
Du 1 juin 2017
au 31 mai 2024
Nutrition and brain health, from predictive biology to disease prevention and treatment - Food4BrainHealth
Programme: Réseau de recherche international (RRI)
Organisme(s) subventionnaire(s): Université Laval - Fonds internes, Université McGill, Université de Toronto, Institut national de la recherche agronomique
Établissement tête: Université Laval
Du 18 mars 2019
au 17 mars 2024
Dissecting host-microbiome modifiers of type 2 diabetes risk - Objective 1.2
Programme: Subvention d'équipe : Initiative canadienne microbiome 2 : Équipes de recherche
Organisme(s) subventionnaire(s): Instituts de recherche en santé du Canada
Établissement tête: Université Laval
Du 1 novembre 2019
au 31 octobre 2024
Dissecting host-microbiome modifiers of type 2 diabetes risk - Objective 1.3
Programme: Subvention d'équipe : Initiative canadienne microbiome 2 : Équipes de recherche
Organisme(s) subventionnaire(s): Instituts de recherche en santé du Canada
Établissement tête: Université Laval
Du 1 novembre 2019
au 31 octobre 2024
Dissecting host-microbiome modifiers of type 2 diabetes risk
Programme: Subvention d'équipe : Initiative canadienne microbiome 2 : Équipes de recherche
Organisme(s) subventionnaire(s): Instituts de recherche en santé du Canada
Établissement tête: Université Laval
Du 1 novembre 2019
au 31 octobre 2024
Dissecting host-microbiome modifiers of type 2 diabetes risk - Objective 1.1
Programme: Subvention d'équipe : Initiative canadienne microbiome 2 : Équipes de recherche
Organisme(s) subventionnaire(s): Instituts de recherche en santé du Canada
Établissement tête: Université Laval
Du 1 novembre 2019
au 31 octobre 2024
Dissecting host-microbiome modifiers of type 2 diabetes risk - Objective 3.2
Programme: Subvention d'équipe : Initiative canadienne microbiome 2 : Équipes de recherche
Organisme(s) subventionnaire(s): Instituts de recherche en santé du Canada
Établissement tête: Université Laval
Du 1 novembre 2019
au 31 octobre 2024
Characterization of the endocannabinoidome of a CDKL5 mouse model
Organisme(s) subventionnaire(s): CDKL5
Établissement tête: Université Laval
Du 15 janvier 2023
au 15 janvier 2024
Effets de lipides polaires laitiers sur l’intégrité intestinale, le système endocannabinoïde et le microbiote fécal chez le porcelet
Programme: Projet subsidiaire d'un regroupement stratégique
Organisme(s) subventionnaire(s): Fonds de recherche du Québec - Nature et technologies
Établissement tête: Université Laval
Du 16 janvier 2023
au 31 mars 2024
Subventions des 5 dernières années
FSAA --- Support de Sentinelle Nord à l'Unité mixte internationale sur la recherche chimique et biomoléculaire de microbiome
Programme: Fonds d'excellence en recherche Apogée Canada
Organisme(s) subventionnaire(s): Secrétariat des programmes interorganismes à l’intention des établissements
Établissement tête: Université Laval
Du 29 novembre 2016
au 31 août 2022
Study of the role of the gut microbiome-endocannabinoidome axis in metabolic health and its therapeutic exploitation
Programme: Fonds des leaders John-R.-Evans (FLJR)
Organisme(s) subventionnaire(s): Ministère de la Santé et des Services sociaux, Ministère de l'éducation et de l'enseignement supérieur, Fondation Canadienne pour l'innovation (La)
Établissement tête: Université Laval
Du 1 avril 2018
au 31 mars 2021
Role of the gut microbiome-endocannabinoidome axis in metabolic health and its therapeutic exploitation - phase 2
Programme: Fonds des leaders John-R.-Evans (FLJR)
Organisme(s) subventionnaire(s): Fondation Canadienne pour l'innovation (La), Ministère de l'éducation et de l'enseignement supérieur
Établissement tête: Université Laval
Du 1 septembre 2018
au 31 mars 2021
The role of full-fat dairy products on body weigth control and metabolic health in adults
Programme: Dairy Research Cluster 3
Organisme(s) subventionnaire(s): Les producteurs laitiers du Canada
Établissement tête: Université Laval
Du 1 septembre 2018
au 31 mars 2023
Aménagement d'espaces de recherche dédiés à de la recherche de pointe sur le microbiome
Programme: Programme de soutien aux organismes de recherche et d'innovation (PSO) - Volet 4: Soutien au financement d'infrastructures de recherche et d'innovation
Organisme(s) subventionnaire(s): Université Laval - Fonds internes, Ministère de l'Économie et de l'Innovation
Établissement tête: Université Laval
Du 1 avril 2019
au 30 novembre 2021
Programme de soutien aux nouveaux chercheurs
Programme: Soutien facultaire aux jeunes chercheurs de la Faculté de médecine
Organisme(s) subventionnaire(s): Université Laval - Fonds internes
Établissement tête: Université Laval
Du 1 juillet 2019
au 30 juin 2022
Territorialiser les systèmes alimentaires : une révolution pour la planète et la santé durable
Organisme(s) subventionnaire(s): Alliance santé Québec (AsQ)
Établissement tête: Université Laval
Du 1 avril 2020
au 31 mars 2021
Microbiome-In-GutVitro: étude préliminaire de séquençage multi-règnes pour le développement d’une approche analytique dans l’identification de microorganismes non-bactériens membres du microbiome intestinal en système M-SHIME
Programme: Projet subsidiaire - Nouveaux Centres et Instituts de recherche - Subventions régulières (pour fins de gestion au VRRCI)
Organisme(s) subventionnaire(s): Fonds de recherche du Québec - Santé
Établissement tête: Université Laval
Du 9 juin 2021
au 8 juin 2022
Supplément de stage - Étude de l'impact de la transplantation fécal sur l'amélioration du diabète après la chirurgie bariatrique
Organisme(s) subventionnaire(s): Sorbonne Université
Établissement tête: Université Laval
Du 5 janvier 2022
au 31 mai 2022
Étude de l'impact de la transplantation fécal sur l'amélioration du diabète après la chirurgie bariatrique
Programme: Réseaux thématiques de recherche
Organisme(s) subventionnaire(s): Fonds de recherche du Québec - Santé
Établissement tête: Université Laval
Du 5 janvier 2022
au 31 mars 2023
Assessment of the direct effects of propolis on the gut microbiome utilizing the Simulator of the Human Intestinal Microbial Ecosystem (SHIME)
Programme: Projet subsidiaire d'un regroupement stratégique
Organisme(s) subventionnaire(s): Fonds de recherche du Québec - Nature et technologies
Établissement tête: Université Laval
Du 1 février 2022
au 31 janvier 2023
Encadrements terminés dans les 5 dernières années
Publications des 5 dernières années
A Lipidomics- and Transcriptomics-Based Analysis of the Intestine of Genetically Obese (ob/ob) and Diabetic (db/db) Mice: Links with Inflammation and Gut Microbiota Cells, 2023/01/25. Francesco Suriano, Claudia Manca, Nicolas Flamand, Matthias Van Hul, Nathalie M. Delzenne, Cristoforo Silvestri, Patrice D. Cani, Vincenzo Di Marzo. DOI 10.3390/cells12030411
The Effects of Peripubertal THC Exposure in Neurodevelopmental Rat Models of Psychopathology International Journal of Molecular Sciences, 2023/02. Martina Di Bartolomeo, Tibor Stark, Serena Di Martino, Fabio Arturo Iannotti, Jana Ruda-Kucerova, Giovanni Luca Romano, Martin Kuchar, Samuele Laudani, Petr Palivec, Fabiana Piscitelli, Carsten T. Wotjak, Claudio Bucolo, Filippo Drago, Vincenzo Di Marzo, claudio d'addario, Vincenzo Micale. DOI 10.3390/ijms24043907
MicroRNA-mediated repression of endocannabinoid CB1 receptor expression contributes to simvastatin-induced skeletal muscle toxicity 2022/12/19. Hilal Kalkan, Elisabetta Panza, Ester Pagano, Giuseppe Ercolano, Claudia Moriello, Fabiana Piscitelli, Raffaele Capasso, Vincenzo Di Marzo, Fabio Iannotti. DOI 10.21203/rs.3.rs-2328769/v1
TRPM8 indicates poor prognosis in colorectal cancer patients and its pharmacological targeting reduces tumour growth in mice by inhibiting Wnt/β-catenin signalling British Journal of Pharmacology, 2023. Pagano, E., Romano, B., Cicia, D., Iannotti, F.A., Venneri, T., Lucariello, G., Nanì, M.F., Cattaneo, F., De Cicco, P., D'Armiento, M., De Luca, M., Lionetti, R., Lama, S., Stiuso, P., Zoppoli, P., Falco, G., Marchianò, S., Fiorucci, S., Capasso, R., Di Marzo, V., Borrelli, F., Izzo, A.A.. DOI 10.1111/bph.15960
Targeting gut dysbiosis against inflammation and impaired autophagy in Duchenne muscular dystrophy EMBO Molecular Medicine, 2023. Kalkan, H., Pagano, E., Paris, D., Panza, E., Cuozzo, M., Moriello, C., Piscitelli, F., Abolghasemi, A., Gazzerro, E., Silvestri, C., Capasso, R., Motta, A., Russo, R., Di Marzo, V., Iannotti, F.A.. DOI 10.15252/emmm.202216225
First Evidence of the Protective Effects of 2-Pentadecyl-2-Oxazoline (PEA-OXA) in In Vitro Models of Acute Lung Injury Biomolecules, 2022/12/24. Aniello Schiano Moriello, Fiorentina Roviezzo, Fabio Arturo Iannotti, Giuseppina Rea, Marco Allarà, Rosa Camerlingo, Roberta Verde, Vincenzo Di Marzo, Stefania Petrosino. DOI 10.3390/biom13010033
Early Blockade of CB1 Receptors Ameliorates Schizophrenia-like Alterations in the Neurodevelopmental MAM Model of Schizophrenia Biomolecules, 2022/01/10. Tibor Stark, Fabio Arturo Iannotti, Serena Di Martino, Martina Di Bartolomeo, Jana Ruda-Kucerova, Fabiana Piscitelli, Carsten T. Wotjak, Claudio D’Addario, Filippo Drago, Vincenzo Di Marzo, Vincenzo Micale. DOI 10.3390/biom12010108
Obesity: The Fat Tissue Disease Version of Cancer Cells, 2022/06/09. Besma Boubertakh, Cristoforo Silvestri, Vincenzo Di Marzo. DOI 10.3390/cells11121872
Mutual Links between the Endocannabinoidome and the Gut Microbiome, with Special Reference to Companion Animals: A Nutritional Viewpoint Animals, 2022/01/31. Aniello Schiano Moriello, Vincenzo Di Marzo, Stefania Petrosino. DOI 10.3390/ani12030348
(Wh)olistic (E)ndocannabinoidome-Microbiome-Axis Modulation through (N)utrition (WHEN) to Curb Obesity and Related Disorders Lipids in Health and Disease, 2022/01/14. Jyoti Sihag, Vincenzo Di Marzo. DOI 10.1186/s12944-021-01609-3
Biosynthesis and metabolism of endocannabinoids and their congeners from the monoacylglycerol and N-acyl-ethanolamine families Biochemical Pharmacology, 2022. Simard, M., Archambault, A.-S., Lavoie, J.-P.C., Dumais, É., Di Marzo, V., Flamand, N.. DOI 10.1016/j.bcp.2022.115261
Adipocyte-specific Nos2 deletion improves insulin resistance and dyslipidemia through brown fat activation in diet-induced obese mice Molecular Metabolism, 2022. Vilela, V.R., Samson, N., Nachbar, R., Perazza, L.R., Lachance, G., Rokatoarivelo, V., Centano-Baez, C., Zancan, P., Sola-Penna, M., Bellmann, K., Di Marzo, V., Laplante, M., Marette, A.. DOI 10.1016/j.molmet.2022.101437
Alterations of the endocannabinoid system and circulating and peripheral tissue levels of endocannabinoids in sarcopenic rats Journal of Cachexia, Sarcopenia and Muscle, 2022. Le Bacquer, O., Salles, J., Piscitelli, F., Sanchez, P., Martin, V., Montaurier, C., Di Marzo, V., Walrand, S.. DOI 10.1002/jcsm.12855
Amygdalar CB2 cannabinoid receptor mediates fear extinction deficits promoted by orexin-A/hypocretin-1 Biomedicine and Pharmacotherapy, 2022. Ten-Blanco, M., Flores, Á., Pereda-Pérez, I., Piscitelli, F., Izquierdo-Luengo, C., Cristino, L., Romero, J., Hillard, C.J., Maldonado, R., Di Marzo, V., Berrendero, F.. DOI 10.1016/j.biopha.2022.112925
Expression and Functions of the CB<sub>2</sub> Receptor in Human Leukocytes Frontiers in Pharmacology, 2022. Simard, M., Rakotoarivelo, V., Di Marzo, V., Flamand, N.. DOI 10.3389/fphar.2022.826400
Cannabinoids and Chronic Liver Diseases International Journal of Molecular Sciences, 2022. Mboumba Bouassa, R.-S., Sebastiani, G., Di Marzo, V., Jenabian, M.-A., Costiniuk, C.T.. DOI 10.3390/ijms23169423
Effects of repeated lysergic acid diethylamide (LSD) on the mouse brain endocannabinoidome and gut microbiome British Journal of Pharmacology, 2022. Inserra, A., Giorgini, G., Lacroix, S., Bertazzo, A., Choo, J., Markopolous, A., Grant, E., Abolghasemi, A., De Gregorio, D., Flamand, N., Rogers, G., Comai, S., Silvestri, C., Gobbi, G., Di Marzo, V.. DOI 10.1111/bph.15977
Exploring the endocannabinoidome in genetically obese (ob/ob) and diabetic (db/db) mice: Links with inflammation and gut microbiota Biochimica et Biophysica Acta - Molecular and Cell Biology of Lipids, 2022. Suriano, F., Manca, C., Flamand, N., Depommier, C., Van Hul, M., Delzenne, N.M., Silvestri, C., Cani, P.D., Di Marzo, V.. DOI 10.1016/j.bbalip.2021.159056
Impact of selenium on the intestinal microbiome-eCBome axis in the context of diet-related metabolic health in mice Frontiers in Immunology, 2022. Guevara Agudelo, F.A., Leblanc, N., Bourdeau-Julien, I., St-Arnaud, G., Lacroix, S., Martin, C., Flamand, N., Veilleux, A., Di Marzo, V., Raymond, F.. DOI 10.3389/fimmu.2022.1028412
Facile and Sustainable Synthesis of Commendamide and its Analogues Frontiers in Chemistry, 2022. Villano, R., Tinto, F., Di Marzo, V.. DOI 10.3389/fchem.2022.858854
Hemp seed significantly modulates the endocannabinoidome and produces beneficial metabolic effects with improved intestinal barrier function and decreased inflammation in mice under a high-fat, high-sucrose diet as compared with linseed Frontiers in Immunology, 2022. Ben Necib, R., Manca, C., Lacroix, S., Martin, C., Flamand, N., Di Marzo, V., Silvestri, C.. DOI 10.3389/fimmu.2022.882455
Human and mouse eosinophils differ in their ability to biosynthesize eicosanoids, docosanoids, the endocannabinoid 2-arachidonoyl-glycerol and its congeners Cells, 2022. Archambault, A.-S., Brassard, J., Bernatchez, É., Martin, C., Di Marzo, V., Laviolette, M., Boulet, L.-P., Blanchet, M.-R., Flamand, N.. DOI 10.3390/cells11010141
Short and efficient synthesis of alkylresorcinols: a route for the preparation of cannabinoids New Journal of Chemistry, 2022. Rosaria Villano, Hannah Straker, Vincenzo Di Marzo. DOI 10.1039/D2NJ03547B
Influence of diet on acute endocannabinoidome mediator levels post exercise in active women, a crossover randomized study Scientific Reports, 2022. Forteza, F., Bourdeau-Julien, I., Nguyen, G.Q., Guevara Agudelo, F.A., Rochefort, G., Parent, L., Rakotoarivelo, V., Feutry, P., Martin, C., Perron, J., Lamarche, B., Flamand, N., Veilleux, A., Billaut, F., Di Marzo, V., Raymond, F.. DOI 10.1038/s41598-022-10757-0
N-Acylethanolamine acid amidase (NAAA) is dysregulated in colorectal cancer patients and its inhibition reduces experimental cancer growth British Journal of Pharmacology, 2022. Romano, B., Pagano, E., Iannotti, F.A., Piscitelli, F., Brancaleone, V., Lucariello, G., Nanì, M.F., Fiorino, F., Sparaco, R., Vanacore, G., Di Tella, F., Cicia, D., Lionetti, R., Makriyannis, A., Malamas, M., De Luca, M., Aprea, G., D'Armiento, M., Capasso, R., Sbarro, B., Venneri, T., Di Marzo, V., Borrelli, F., Izzo, A.A.. DOI 10.1111/bph.15737
Positive association between plasmatic levels of orexin A and the endocannabinoid-derived 2-arachidonoyl lysophosphatidic acid in Alzheimer’s disease Frontiers in Aging Neuroscience, 2022. Forte, N., Fernández-Rilo, A.C., Palomba, L., Marfella, B., Piscitelli, F., De Girolamo, P., Di Costanzo, A., Di Marzo, V., Cristino, L.. DOI 10.3389/fnagi.2022.1004002
Cannabinoids: a class of unique natural products with unique pharmacology Rendiconti Lincei. Scienze Fisiche e Naturali, 2021/03/11. Fabiana Piscitelli, Vincenzo Di Marzo. DOI 10.1007/s12210-020-00966-y
Short-term supplementation with ω-3 polyunsaturated fatty acids modulates primarily mucolytic species from the gut luminal mucin niche in a human fermentation system Gut Microbes, 2022. Roussel, C., Anunciação Braga Guebara, S., Plante, P.-L., Desjardins, Y., Di Marzo, V., Silvestri, C.. DOI 10.1080/19490976.2022.2120344
The endocannabinoidome mediator N-oleoylglycine is a novel protective agent against 1-methyl-4-phenyl-pyridinium-induced neurotoxicity Frontiers in Aging Neuroscience, 2022. Lauritano, A., Cipollone, I., Verde, R., Kalkan, H., Moriello, C., Iannotti, F.A., Di Marzo, V., Piscitelli, F.. DOI 10.3389/fnagi.2022.926634
Three of a kind: Control of the expression of liver-expressed antimicrobial peptide 2 (leap2) by the endocannabinoidome and the gut microbiome Molecules, 2022. Shen, M., Manca, C., Suriano, F., Nallabelli, N., Pechereau, F., Allam-Ndoul, B., Iannotti, F.A., Flamand, N., Veilleux, A., Cani, P.D., Silvestri, C., Di Marzo, V.. DOI 10.3390/molecules27010001
Assessment of the effects of dietary vitamin d levels on olanzapine-induced metabolic side effects: Focus on the endocannabinoidome-gut microbiome axis International Journal of Molecular Sciences, 2021. Abolghasemi, A., Manca, C., Iannotti, F.A., Shen, M., Leblanc, N., Lacroix, S., Martin, C., Flamand, N., Di Marzo, V., Silvestri, C.. DOI 10.3390/ijms222212361
A Glucuronic Acid-Palmitoylethanolamide Conjugate (GLUPEA) Is an Innovative Drug Delivery System and a Potential Bioregulator Cells, 2021/02/20. Emiliano Manzo, Aniello Schiano Moriello, Francesco Tinto, Roberta Verde, Marco Allarà, Luciano De Petrocellis, Ester Pagano, Angelo A. Izzo, Vincenzo Di Marzo, Stefania Petrosino. DOI 10.3390/cells10020450
Linking the Endocannabinoidome with Specific Metabolic Parameters in an Overweight and Insulin-Resistant Population: From Multivariate Exploratory Analysis to Univariate Analysis and Construction of Predictive Models Cells, 2021/01/05. Clara Depommier, Nicolas Flamand, Rudy Pelicaen, Dominique Maiter, Jean-Paul Thissen, Audrey Loumaye, Michel P. Hermans, Amandine Everard, Nathalie M. Delzenne, Vincenzo Di Marzo, Patrice D. Cani. DOI 10.3390/cells10010071
2-Pentadecyl-2-oxazoline ameliorates memory impairment and depression-like behaviour in neuropathic mice: possible role of adrenergic alpha2- and H3 histamine autoreceptors Molecular Brain, 2021. Boccella, S., Guida, F., Iannotta, M., Iannotti, F.A., Infantino, R., Ricciardi, F., Cristiano, C., Vitale, R.M., Amodeo, P., Marabese, I., Belardo, C., de Novellis, V., Paino, S., Palazzo, E., Calignano, A., Di Marzo, V., Maione, S., Luongo, L.. DOI 10.1186/s13041-020-00724-z
Correction to: 2-Pentadecyl-2-oxazoline ameliorates memory impairment and depression-like behaviour in neuropathic mice: possible role of adrenergic alpha2- and H3 histamine autoreceptors (Molecular Brain, (2021), 14, 1, (28), 10.1186/s13041-020-00724-z) Molecular Brain, 2021. Boccella, S., Guida, F., Iannotta, M., Iannotti, F.A., Infantino, R., Ricciardi, F., Cristiano, C., Vitale, R.M., Amodeo, P., Marabese, I., Belardo, C., de Novellis, V., Paino, S., Palazzo, E., Calignano, A., Di Marzo, V., Maione, S., Luongo, L.. DOI 10.1186/s13041-021-00772-z
B iological basis of cannabinoid medicines: Mechanistic insights into cannabinoid signaling could improve therapeutic applications Science, 2021. Keimpema, E., Marzo, V.D., Harkany, T.. DOI 10.1126/science.abf6099
Beneficial effects of akkermansia muciniphila are not associated with major changes in the circulating endocannabinoidome but linked to higher mono-palmitoyl-glycerol levels as new pparα agonists Cells, 2021. Depommier, C., Vitale, R.M., Iannotti, F.A., Silvestri, C., Flamand, N., Druart, C., Everard, A., Pelicaen, R., Maiter, D., Thissen, J.-P., Loumaye, A., Hermans, M.P., Delzenne, N.M., de Vos, W.M., Marzo, V.D., Cani, P.D.. DOI 10.3390/cells10010185
Biosynthesis of the novel endogenous 15-lipoxygenase metabolites N-13-hydroxy-octodecadienoyl-ethanolamine and 13-hydroxy-octodecadienoyl-glycerol by human neutrophils and Eosinophils Cells, 2021. Archambault, A.-S., Tinto, F., Dumais, É., Rakotoarivelo, V., Kostrzewa, M., Plante, P.-L., Martin, C., Simard, M., Silvestri, C., Pouliot, R., Laviolette, M., Boulet, L.-P., Vitale, R.M., Ligresti, A., Di Marzo, V., Flamand, N.. DOI 10.3390/cells10092322
Effect of docosahexaenoic acid (DHA) at the enteric level in a synucleinopathy mouse model Nutrients, 2021. Lamontagne‐proulx, J., Coulombe, K., Dahhani, F., Côté, M., Guyaz, C., Tremblay, C., Di Marzo, V., Flamand, N., Calon, F., Soulet, D.. DOI 10.3390/nu13124218
Crosstalk between the transcriptional regulation of dopamine D2 and cannabinoid CB1 receptors in schizophrenia: Analyses in patients and in perinatal Δ9-tetrahydrocannabinol-exposed rats Pharmacological Research, 2021. Di Bartolomeo, M., Stark, T., Maurel, O.M., Iannotti, F.A., Kuchar, M., Ruda-Kucerova, J., Piscitelli, F., Laudani, S., Pekarik, V., Salomone, S., Arosio, B., Mechoulam, R., Maccarrone, M., Drago, F., Wotjak, C.T., Di Marzo, V., Vismara, M., Dell'Osso, B., D'Addario, C., Micale, V.. DOI 10.1016/j.phrs.2020.105357
Deletion of the gene encoding prostamide/prostaglandin F synthase reveals an important role in regulating intraocular pressure Prostaglandins Leukotrienes and Essential Fatty Acids, 2021. Bertrand, J.A., Woodward, D.F., Sherwood, J.M., Spenlehauer, A., Silvestri, C., Piscitelli, F., Marzo, V.D., Yamazaki, M., Sakimura, K., Inoue, Y., Watanabe, K., Overby, D.R.. DOI 10.1016/j.plefa.2020.102235
Editorial on “Cannabis and cannabinoids: history, practice and socio-economical inferences of a controversial plant” Rendiconti Lincei, 2021. Di Marzo, V., Marino, G.. DOI 10.1007/s12210-021-00975-5
Intuitive eating is associated with elevated levels of circulating omega-3-polyunsaturated fatty acid-derived endocannabinoidome mediators Appetite, 2021. Rochefort, G., Provencher, V., Castonguay-Paradis, S., Perron, J., Lacroix, S., Martin, C., Flamand, N., Di Marzo, V., Veilleux, A.. DOI 10.1016/j.appet.2020.104973
Efficacy of combined therapy with fish oil and phytocannabinoids in murine intestinal inflammation Phytotherapy Research, 2021. Pagano, E., Iannotti, F.A., Piscitelli, F., Romano, B., Lucariello, G., Venneri, T., Di Marzo, V., Izzo, A.A., Borrelli, F.. DOI 10.1002/ptr.6831
Genetic Manipulation of sn-1-Diacylglycerol Lipase and CB<sub>1</sub>Cannabinoid Receptor Gain-of-Function Uncover Neuronal 2-Linoleoyl Glycerol Signaling in Drosophila melanogaster Cannabis and Cannabinoid Research, 2021. Tortoriello, G., Beiersdorf, J., Romani, S., Williams, G., Cameron, G.A., Mackie, K., Williams, M.J., Di Marzo, V., Keimpema, E., Doherty, P., Harkany, T.. DOI 10.1089/can.2020.0010
Identification and characterization of cannabidiol as an ox1r antagonist by computational and in vitro functional validation Biomolecules, 2021. Vitale, R.M., Iannotti, F.A., Moriello, A.S., Tunisi, L., Piscitelli, F., Savopoulos, R., Cristino, L., De Petrocellis, L., Amodeo, P., Gray, R., Di Marzo, V.. DOI 10.3390/biom11081134
N-palmitoyl-d-glucosamine, a natural monosaccharide-based glycolipid, inhibits tlr4 and prevents lps-induced inflammation and neuropathic pain in mice International Journal of Molecular Sciences, 2021. Iannotta, M., Belardo, C., Trotta, M.C., Iannotti, F.A., Vitale, R.M., Maisto, R., Boccella, S., Infantino, R., Ricciardi, F., Mirto, B.F., Ferraraccio, F., Panarese, I., Amodeo, P., Tunisi, L., Cristino, L., D’amico, M., Di Marzo, V., Luongo, L., Maione, S., Guida, F.. DOI 10.3390/ijms22031491
Kahweol, a natural diterpene from coffee, induces peripheral antinociception by endocannabinoid system activation Brazilian Journal of Medical and Biological Research, 2021. L.S. Guzzo, C.C. Oliveira, R.C.M. Ferreira, D.P.D. Machado, M.G.M. Castor, A.C. Perez, F. Piscitelli, V. Di Marzo, T.R.L. Romero, I.D.G. Duarte. DOI 10.1590/1414-431x2021e11071
Maternal omega-3 intake differentially affects the endocannabinoid system in the progeny`s neocortex and hippocampus: Impact on synaptic markers Journal of Nutritional Biochemistry, 2021. Isaac, A.R., de Velasco, P.C., Fraga, K.Y.D., Tavares-do-Carmo, M.D.G., Campos, R.M.P., Iannotti, F.A., Verde, R., Martins, D.B.G., Santos, T.A., Ferreira, B.K., de Mello, F.G., Di Marzo, V., Andrade-da-Costa, B.L.D.S., de Melo Reis, R.A.. DOI 10.1016/j.jnutbio.2021.108782
N-Oleoylglycine and N-Oleoylalanine Do Not Modify Tolerance to Nociception, Hyperthermia, and Suppression of Activity Produced by Morphine Frontiers in Synaptic Neuroscience, 2021. Rock, E.M., Limebeer, C.L., Sullivan, M.T., DeVuono, M.V., Lichtman, A.H., Di Marzo, V., Mechoulam, R., Parker, L.A.. DOI 10.3389/fnsyn.2021.620145
Spontaneous and Naloxone-Precipitated Withdrawal Behaviors From Chronic Opiates are Accompanied by Changes in N-Oleoylglycine and N-Oleoylalanine Levels in the Brain and Ameliorated by Treatment With These Mediators Frontiers in Pharmacology, 2021. Ayoub, S.M., Piscitelli, F., Silvestri, C., Limebeer, C.L., Rock, E.M., Smoum, R., Farag, M., de Almeida, H., Sullivan, M.T., Lacroix, S., Boubertakh, B., Nallabelli, N., Lichtman, A.H., Leri, F., Mechoulam, R., Di Marzo, V., Parker, L.A.. DOI 10.3389/fphar.2021.706703
Oral capsaicinoid administration alters the plasma endocannabinoidome and fecal microbiota of reproductive-aged women living with overweight and obesity Biomedicines, 2021. Manca, C., Lacroix, S., Pérusse, F., Flamand, N., Chagnon, Y., Drapeau, V., Tremblay, A., Di Marzo, V., Silvestri, C.. DOI 10.3390/biomedicines9091246
Orexin-A and endocannabinoids are involved in obesity-associated alteration of hippocampal neurogenesis, plasticity, and episodic memory in mice Nature Communications, 2021. Forte, N., Boccella, S., Tunisi, L., Fernández-Rilo, A.C., Imperatore, R., Iannotti, F.A., De Risi, M., Iannotta, M., Piscitelli, F., Capasso, R., De Girolamo, P., De Leonibus, E., Maione, S., Di Marzo, V., Cristino, L.. DOI 10.1038/s41467-021-26388-4
Orexin-A/Hypocretin-1 Controls the VTA-NAc Mesolimbic Pathway via Endocannabinoid-Mediated Disinhibition of Dopaminergic Neurons in Obese Mice Frontiers in Synaptic Neuroscience, 2021. Tunisi, L., D'Angelo, L., Fernández-Rilo, A.C., Forte, N., Piscitelli, F., Imperatore, R., de Girolamo, P., Di Marzo, V., Cristino, L.. DOI 10.3389/fnsyn.2021.622405
Role of 2-Arachidonoyl-Glycerol and CB1 Receptors in Orexin-A-Mediated Prevention of Oxygen–Glucose Deprivation-Induced Neuronal Injury Cells, 2020/06/20. Letizia Palomba, Andrea Motta, Roberta Imperatore, Fabiana Piscitelli, Raffaele Capasso, Federica Mastroiacovo, Giuseppe Battaglia, Valeria Bruno, Luigia Cristino, Vincenzo Di Marzo. DOI 10.3390/cells9061507
Synthesis and molecular targets of N-13-hydroxy-octadienoyl-ethanolamine, a novel endogenous bioactive 15-lipoxygenase-derived metabolite of N-linoleoyl-ethanolamine found in the skin and saliva Biochimica et Biophysica Acta - Molecular and Cell Biology of Lipids, 2021. Tinto, F., Archambault, A.-S., Dumais, É., Rakotoarivelo, V., Kostrzewa, M., Martin, C., Plante, P.-L., Desjardins, Y., Simard, M., Pouliot, R., De Petrocellis, L., Ligresti, A., Di Marzo, V., Flamand, N.. DOI 10.1016/j.bbalip.2021.158954
The gut microbiome, endocannabinoids and metabolic disorders Journal of Endocrinology, 2021. Iannotti, F.A., Di Marzo, V.. DOI 10.1530/JOE-20-0444
Mgll Knockout Mouse Resistance to Diet-Induced Dysmetabolism Is Associated with Altered Gut Microbiota Cells, 2020/12/17. Niokhor Dione, Sébastien Lacroix, Ulrike Taschler, Thomas Deschênes, Armita Abolghasemi, Nadine Leblanc, Vincenzo Di Marzo, Cristoforo Silvestri. DOI 10.3390/cells9122705
Acute naloxone-precipitated morphine withdrawal elicits nausea-like somatic behaviors in rats in a manner suppressed by N-oleoylglycine Psychopharmacology, 2020. Rock, E.M., Ayoub, S.M., Limebeer, C.L., Gene, A., Wills, K.L., DeVuono, M.V., Smoum, R., Di Marzo, V., Lichtman, A.H., Mechoulam, R., Parker, L.A.. DOI 10.1007/s00213-019-05373-2
Hepatic NAPE-PLD Is a Key Regulator of Liver Lipid Metabolism Cells, 2020/05/18. Charlotte Lefort, Martin Roumain, Matthias Van Hul, Marialetizia Rastelli, Rita Manco, Isabelle Leclercq, Nathalie M. Delzenne, Vincenzo Di Marzo, Nicolas Flamand, Serge Luquet, Cristoforo Silvestri, Giulio G. Muccioli, Patrice D. Cani. DOI 10.3390/cells9051247
Obesity Affects the Microbiota–Gut–Brain Axis and the Regulation Thereof by Endocannabinoids and Related Mediators International Journal of Molecular Sciences, 2020/02/25. Nicola Forte, Alba Clara Fernández-Rilo, Letizia Palomba, Vincenzo Di Marzo, Luigia Cristino. DOI 10.3390/ijms21051554
Cannabinoids and the expanded endocannabinoid system in neurological disorders Nature Reviews Neurology, 2020/01. Luigia Cristino, Tiziana Bisogno, Vincenzo Di Marzo. DOI 10.1038/s41582-019-0284-z
Anticonvulsive Properties of Cannabidiol in a Model of Generalized Seizure Are Transient Receptor Potential Vanilloid 1 Dependent Cannabis and Cannabinoid Research, 2020. Gray, R.A., Stott, C.G., Jones, N.A., Di Marzo, V., Di Marzo, V., Whalley, B.J., Whalley, B.J.. DOI 10.1089/can.2019.0028
Adverse effects of Δ<sup>9</sup>-tetrahydrocannabinol on neuronal bioenergetics during postnatal development JCI Insight, 2020. Beiersdorf, J., Hevesi, Z., Calvigioni, D., Pyszkowski, J., Romanov, R., Szodorai, E., Lubec, G., Shirran, S., Botting, C.H., Kasper, S., Guy, G.W., Gray, R., Marzo, V.D., Harkany, T., Keimpema, E.. DOI 10.1172/jci.insight.135418
Alterations of brain endocannabinoidome signaling in germ-free mice Biochimica et Biophysica Acta - Molecular and Cell Biology of Lipids, 2020. Manca, C., Shen, M., Boubertakh, B., Martin, C., Flamand, N., Silvestri, C., Di Marzo, V.. DOI 10.1016/j.bbalip.2020.158786
Altered dopamine D3 receptor gene expression in MAM model of schizophrenia is reversed by peripubertal cannabidiol treatment Biochemical Pharmacology, 2020. Stark, T., Di Bartolomeo, M., Di Marco, R., Drazanova, E., Platania, C.B.M., Iannotti, F.A., Ruda-Kucerova, J., D'Addario, C., Kratka, L., Pekarik, V., Piscitelli, F., Babinska, Z., Fedotova, J., Giurdanella, G., Salomone, S., Sulcova, A., Bucolo, C., Wotjak, C.T., Starcuk, Z., Drago, F., Mechoulam, R., Di Marzo, V., Micale, V.. DOI 10.1016/j.bcp.2020.114004
Design, Synthesis and In Vitro Experimental Validation of Novel TRPV4 Antagonists Inspired by Labdane Diterpenes Marine drugs, 2020. Mazzotta, S., Carullo, G., Schiano Moriello, A., Amodeo, P., Di Marzo, V., Vega-Holm, M., Vitale, R.M., Aiello, F., Brizzi, A., De Petrocellis, L.. DOI 10.3390/md18100519
Cannabidiol in sport: Ergogenic or else? Pharmacological Research, 2020. Gamelin, F.-X., Cuvelier, G., Mendes, A., Aucouturier, J., Berthoin, S., Di Marzo, V., Heyman, E.. DOI 10.1016/j.phrs.2020.104764
Comments on Disruption of the gonadal endocannabinoid system in zebrafish exposed to diisononyl phthalate – Forner-Piquer et al. (2018)”: rebuttal to Prosser CM. Environmental Pollution, 2020. Forner-Piquer, I., Santangeli, S., Maradonna, F., Rabbito, A., Piscitelli, F., Habibi, H.R., di Marzo, V., Carnevali, O.. DOI 10.1016/j.envpol.2020.114028
Desensitization of transient receptor potential vanilloid type-1 (TRPV1) channel as promising therapy of irritable bowel syndrome: characterization of the action of palvanil in the mouse gastrointestinal tract Naunyn-Schmiedeberg's Archives of Pharmacology, 2020. Szymaszkiewicz, A., Włodarczyk, J., Wasilewski, A., Di Marzo, V., Storr, M., Fichna, J., Zielińska, M.. DOI 10.1007/s00210-020-01829-x
Endocannabinoid hydrolysis inhibition unmasks that unsaturated fatty acids induce a robust biosynthesis of 2-arachidonoyl-glycerol and its congeners in human myeloid leukocytes FASEB Journal, 2020. Turcotte, C., Archambault, A.-S., Dumais, É., Martin, C., Blanchet, M.-R., Bissonnette, E., Ohashi, N., Yamamoto, K., Itoh, T., Laviolette, M., Veilleux, A., Boulet, L.-P., Di Marzo, V., Flamand, N.. DOI 10.1096/fj.201902916R
Design, Synthesis, and Physicochemical and Pharmacological Profiling of 7-Hydroxy-5-oxopyrazolo[4,3-b]pyridine-6-carboxamide Derivatives with Antiosteoarthritic Activity in Vivo Journal of Medicinal Chemistry, 2020. Mugnaini, C., Kostrzewa, M., Bryk, M., Mahmoud, A.M., Brizzi, A., Lamponi, S., Giorgi, G., Ferlenghi, F., Vacondio, F., MacCioni, P., Colombo, G., Mor, M., Starowicz, K., Di Marzo, V., Ligresti, A., Corelli, F.. DOI 10.1021/acs.jmedchem.0c00595
Dietary fatty acid intake and gut microbiota determine circulating endocannabinoidome signaling beyond the effect of body fat Scientific Reports, 2020. Castonguay-Paradis, S., Lacroix, S., Rochefort, G., Parent, L., Perron, J., Martin, C., Lamarche, B., Raymond, F., Flamand, N., Di Marzo, V., Veilleux, A.. DOI 10.1038/s41598-020-72861-3
Effects of BPA on zebrafish gonads: Focus on the endocannabinoid system Environmental Pollution, 2020. Forner-Piquer, I., Beato, S., Piscitelli, F., Santangeli, S., Di Marzo, V., Habibi, H.R., Maradonna, F., Carnevali, O.. DOI 10.1016/j.envpol.2020.114710
Germ-free mice exhibit profound gut microbiota-dependent alterations of intestinal endocannabinoidome signaling Journal of Lipid Research, 2020. Manca, C., Boubertakh, B., Leblanc, N., Deschênes, T., Lacroix, S., Martin, C., Houde, A., Veilleux, A., Flamand, N., Muccioli, G.G., Raymond, F., Cani, P.D., Di Marzo, V., Silvestri, C.. DOI 10.1194/jlr.RA119000424
Erratum: Correction to Design, Synthesis, and Physicochemical and Pharmacological Profiling of 7-Hydroxy-5-oxopyrazolo[4,3- b]pyridine-6-carboxamide Derivatives with Antiosteoarthritic Activity in Vivo (Journal of Medicinal Chemistry (2020) 63:(13);7369-7391. (DOI: 10.1021/acs.jmedchem.0c00595) Journal of Medicinal Chemistry, 2020. Mugnaini, C., Kostrzewa, M., Bryk, M., Mahmoud, A.M., Brizzi, A., Lamponi, S., Giorgi, G., Ferlenghi, F., Vacondio, F., Maccioni, P., Colombo, G., Mor, M., Starowicz, K., Di Marzo, V., Ligresti, A., Corelli, F.. DOI 10.1021/acs.jmedchem.0c01567
Fish Oil, Cannabidiol and the Gut Microbiota: An Investigation in a Murine Model of Colitis Frontiers in Pharmacology, 2020. Silvestri, C., Pagano, E., Lacroix, S., Venneri, T., Cristiano, C., Calignano, A., Parisi, O.A., Izzo, A.A., Di Marzo, V., Borrelli, F.. DOI 10.3389/fphar.2020.585096
Gene deletion studies reveal a critical role for prostamide/prostaglandin F2α synthase in prostamide f2α formation bioRxiv, 2020. Bertrand, J.A., Woodward, D.F., Sherwood, J.M., Spenlehauer, A., Silvestri, C., Piscitelli, F., Di Marzo, V., Yamazaki, M., Sakimura, K., Watanabe, K., Overby, D.R.. DOI 10.1101/2020.04.01.020768
Phytocannabinoids promote viability and functional adipogenesis of bone marrow-derived mesenchymal stem cells through different molecular targets Biochemical Pharmacology, 2020. Fellous, T., De Maio, F., Kalkan, H., Carannante, B., Boccella, S., Petrosino, S., Maione, S., Di Marzo, V., Iannotti, F.A.. DOI 10.1016/j.bcp.2020.113859
Life-long epigenetic programming of cortical architecture by maternal ‘Western’ diet during pregnancy Molecular Psychiatry, 2020. Cinquina, V., Calvigioni, D., Farlik, M., Halbritter, F., Fife-Gernedl, V., Shirran, S.L., Fuszard, M.A., Botting, C.H., Poullet, P., Piscitelli, F., Máté, Z., Szabó, G., Yanagawa, Y., Kasper, S., Di Marzo, V., Mackie, K., McBain, C.J., Bock, C., Keimpema, E., Harkany, T.. DOI 10.1038/s41380-019-0580-4
Manipulation of dietary amino acids prevents and reverses obesity in mice through multiple mechanisms that modulate energy homeostasis Diabetes, 2020. Ruocco, C., Ragni, M., Rossi, F., Carullo, P., Ghini, V., Piscitelli, F., Cutignano, A., Manzo, E., Ioris, R.M., Bontems, F., Tedesco, L., Greco, C.M., Pino, A., Severi, I., Liu, D., Ceddia, R.P., Ponzoni, L., Tenori, L., Rizzetto, L., Scholz, M., Tuohy, K., Bifari, F., Di Marzo, V., Luchinat, C., Carruba, M.O., Cinti, S., Decimo, I., Condorelli, G., Coppari, R., Collins, S., Valerio, A., Nisoli, E.. DOI 10.2337/db20-0489
Oleoyl alanine (HU595): a stable monomethylated oleoyl glycine interferes with acute naloxone precipitated morphine withdrawal in male rats Psychopharmacology, 2020. Ayoub, S.M., Smoum, R., Farag, M., Atwal, H., Collins, S.A., Rock, E.M., Limebeer, C.L., Piscitelli, F., Iannotti, F.A., Lichtman, A.H., Leri, F., Di Marzo, V., Mechoulam, R., Parker, L.A.. DOI 10.1007/s00213-020-05570-4
Treatment With 2-Pentadecyl-2-Oxazoline Restores Mild Traumatic Brain Injury-Induced Sensorial and Neuropsychiatric Dysfunctions Frontiers in Pharmacology, 2020. Boccella, S., Iannotta, M., Cristiano, C., Iannotti, F.A., Bello, F.D., Guida, F., Belardo, C., Infantino, R., Ricciardi, F., Giannella, M., Calignano, A., Di Marzo, V., Maione, S., Luongo, L.. DOI 10.3389/fphar.2020.00091
Protective Effects of N-Oleoylglycine in a Mouse Model of Mild Traumatic Brain Injury ACS Chemical Neuroscience, 2020. Piscitelli, F., Guida, F., Luongo, L., Iannotti, F.A., Boccella, S., Verde, R., Lauritano, A., Imperatore, R., Smoum, R., Cristino, L., Lichtman, A.H., Parker, L.A., Mechoulam, R., Maione, S., Di Marzo, V.. DOI 10.1021/acschemneuro.9b00633
Synthetic bioactive olivetol-related amides: The influence of the phenolic group in cannabinoid receptor activity Bioorganic and Medicinal Chemistry, 2020. Brizzi, A., Aiello, F., Boccella, S., Cascio, M.G., De Petrocellis, L., Frosini, M., Gado, F., Ligresti, A., Luongo, L., Marini, P., Mugnaini, C., Pessina, F., Corelli, F., Maione, S., Manera, C., Pertwee, R.G., Di Marzo, V.. DOI 10.1016/j.bmc.2020.115513
The endocannabinoidome as a substrate for noneuphoric phytocannabinoid action and gut microbiome dysfunction in neuropsychiatric disorders Dialogues in Clinical Neuroscience, 2020. Di Marzo, V.. DOI 10.31887/DCNS.2020.22.3/VDIMARZO
Effects of Dietary Bisphenol A on the Reproductive Function of Gilthead Sea Bream (Sparus aurata) Testes International Journal of Molecular Sciences, 2019/10/10. Isabel Forner-Piquer, Ioannis Fakriadis, Constantinos C Mylonas, Fabiana Piscitelli, Vincenzo Di Marzo, Francesca Maradonna, Josep Calduch-Giner, Jaume Pérez-Sánchez, Oliana Carnevali. DOI 10.3390/ijms20205003
α<sub>2</sub>-Adrenoceptor agonist induces peripheral antinociception via the endocannabinoid system Pharmacological Reports, 2020. Romero, T.R.L., Miranda e Castor, M.G., Parrella, C., Piscitelli, F., Di Marzo, V., Duarte, I.D.G.. DOI 10.1007/s43440-019-00053-6
Cannabidiol improves vocal learning-dependent recovery from, and reduces magnitude of deficits following, damage to a cortical-like brain region in a songbird pre-clinical animal model Neuropharmacology, 2019/11. Ali Alalawi, Julien C. Dodu, Marie Woolley-Roberts, James Brodie, Vincenzo Di Marzo, Ken Soderstrom. DOI 10.1016/j.neuropharm.2019.107716
Corrigendum to “Systemic administration of serotonin exacerbates abdominal pain and colitis via interaction with the endocannabinoid system” [Biochem. Pharmacol. 161 (2019) 37–51] Biochemical Pharmacology, 2019/11. Maciej Salaga, Agata Binienda, Fabiana Piscitelli, Anna Mokrowiecka, Adam I. Cygankiewicz, Roberta Verde, Ewa Malecka-Panas, Radzislaw Kordek, Wanda M. Krajewska, Vincenzo Di Marzo, Jakub Fichna. DOI 10.1016/j.bcp.2019.113636
Human leukocytes differentially express endocannabinoid‐glycerol lipases and hydrolyze 2‐arachidonoyl‐glycerol and its metabolites from the 15‐lipoxygenase and cyclooxygenase pathways Journal of Leukocyte Biology, 2019/09. Caroline Turcotte, Élizabeth Dumais, Anne‐Sophie Archambault, Cyril Martin, Marie‐Renée Blanchet, Élyse Bissonnette, Louis‐Philippe Boulet, Michel Laviolette, Vincenzo Di Marzo, Nicolas Flamand. DOI 10.1002/jlb.3a0919-049rrr
Structure-activity relationships of thiazole and benzothiazole derivatives as selective cannabinoid CB2 agonists with in vivo anti-inflammatory properties European Journal of Medicinal Chemistry, 2019/10. Aya E. Ghonim, Alessia Ligresti, Alessandro Rabbito, Ali Mokhtar Mahmoud, Vincenzo Di Marzo, Noha A. Osman, Ashraf H. Abadi. DOI 10.1016/j.ejmech.2019.07.002
Cannabinoid receptors (version 2019.4) in the IUPHAR/BPS Guide to Pharmacology Database IUPHAR/BPS Guide to Pharmacology CITE, 2019/09/16. Mary Abood, Stephen P.H. Alexander, Francis Barth, Tom I. Bonner, Heather Bradshaw, Guy Cabral, Pierre Casellas, Ben F. Cravatt, William A. Devane, Vincenzo Di Marzo, Maurice R. Elphick, Christian C. Felder, Peter Greasley, Miles Herkenham, Allyn C. Howlett, George Kunos, Ken Mackie, Raphael Mechoulam, Roger G. Pertwee, Ruth A. Ross. DOI 10.2218/gtopdb/F13/2019.4
Discovery of novel benzofuran-based compounds with neuroprotective and immunomodulatory properties for Alzheimer's disease treatment European Journal of Medicinal Chemistry, 2019/09. Serena Montanari, Ali Mokhtar Mahmoud, Letizia Pruccoli, Alessandro Rabbito, Marina Naldi, Sabrina Petralla, Ignacio Moraleda, Manuela Bartolini, Barbara Monti, Isabel Iriepa, Federica Belluti, Silvia Gobbi, Vincenzo Di Marzo, Alessandra Bisi, Andrea Tarozzi, Alessia Ligresti, Angela Rampa. DOI 10.1016/j.ejmech.2019.05.080
Targeted Lipidomics Investigation of N ‐acylethanolamines in a Transgenic Mouse Model of AD: A Longitudinal Study European Journal of Lipid Science and Technology, 2019/07. Fabiana Piscitelli, Roberto Coccurello, Antonio Totaro, Alessandro Leuti, Giacomo Giacovazzo, Roberta Verde, Emanuela Rossi, Michele Podaliri Vulpiani, Nicola Ferri, Roberto Giacominelli Stuffler, Vincenzo Di Marzo, Sergio Oddi, Tiziana Bisogno, Mauro Maccarrone. DOI 10.1002/ejlt.201900015
The non-euphoric phytocannabinoid cannabidivarin counteracts intestinal inflammation in mice and cytokine expression in biopsies from UC pediatric patients Pharmacological Research, 2019/09. E. Pagano, B. Romano, F.A. Iannotti, O.A. Parisi, M. D’Armiento, S. Pignatiello, L. Coretti, M. Lucafò, T. Venneri, G. Stocco, F. Lembo, P. Orlando, R. Capasso, V. Di Marzo, A.A. Izzo, F. Borrelli. DOI 10.1016/j.phrs.2019.104464
Lifestyle and Metabolic Syndrome: Contribution of the Endocannabinoidome Nutrients, 2019/08. Vincenzo Di Marzo, Cristoforo Silvestri. DOI 10.3390/nu11081956
Altered Metabolism of Phospholipases, Diacylglycerols, Endocannabinoids, and N-Acylethanolamines in Patients with Mastocytosis Journal of Immunology Research, 2019/07/01. Anne Lise Ferrara, Fabiana Piscitelli, Angelica Petraroli, Roberta Parente, Maria Rosaria Galdiero, Gilda Varricchi, Giancarlo Marone, Massimo Triggiani, Vincenzo Di Marzo, Stefania Loffredo. DOI 10.1155/2019/5836476
N-Oleoyl-glycine reduces nicotine reward and withdrawal in mice Neuropharmacology, 2019/04. Giulia Donvito, Fabiana Piscitelli, Pretal Muldoon, Asti Jackson, Rosa Maria Vitale, Enrico D'Aniello, Catia Giordano, Bogna M. Ignatowska-Jankowska, Mohammed A. Mustafa, Francesca Guida, Gavin N. Petrie, Linda Parker, Reem Smoum, Laura Sim-Selley, Sabatino Maione, Aron H. Lichtman, M. Imad Damaj, Vincenzo Di Marzo, Raphael Mechoulam. DOI 10.1016/j.neuropharm.2018.03.020
Cannabidivarin completely rescues cognitive deficits and delays neurological and motor defects in male Mecp2 mutant mice Journal of Psychopharmacology, 2019/05. Erica Zamberletti, Marina Gabaglio, Fabiana Piscitelli, James S Brodie, Marie Woolley-Roberts, Isabella Barbiero, Marco Tramarin, Giorgio Binelli, Nicoletta Landsberger, Charlotte Kilstrup-Nielsen, Tiziana Rubino, Vincenzo Di Marzo, Daniela Parolaro. DOI 10.1177/0269881119844184
Orexin-A Prevents Lipopolysaccharide-Induced Neuroinflammation at the Level of the Intestinal Barrier Frontiers in Endocrinology, 2019/04/10. Lea Tunisi, Nicola Forte, Alba Clara Fernández-Rilo, Isabella Mavaro, Raffaele Capasso, Livia D'Angelo, Nataša Milić, Luigia Cristino, Vincenzo Di Marzo, Letizia Palomba. DOI 10.3389/fendo.2019.00219
Altered gut microbiota and endocannabinoid system tone in vitamin D deficiency-mediated chronic pain Brain, Behavior, and Immunity, 2019/04. Francesca Guida, Serena Boccella, Carmela Belardo, Monica Iannotta, Fabiana Piscitelli, Francesca De Filippis, Salvatore Paino, Flavia Ricciardi, Dario Siniscalco, Ida Marabese, Livio Luongo, Danilo Ercolini, Vincenzo Di Marzo, Sabatino Maione. DOI 10.1016/j.bbi.2019.04.006
Systemic administration of serotonin exacerbates abdominal pain and colitis via interaction with the endocannabinoid system Biochemical Pharmacology, 2019/03. Maciej Salaga, Agata Binienda, Fabiana Piscitelli, Anna Mokrowiecka, Adam I. Cygankiewicz, Roberta Verde, Ewa Malecka-Panas, Radzislaw Kordek, Wanda M. Krajewska, Vincenzo Di Marzo, Jakub Fichna. DOI 10.1016/j.bcp.2019.01.001
Oleoyl glycine: interference with the aversive effects of acute naloxone-precipitated MWD, but not morphine reward, in male Sprague–Dawley rats Psychopharmacology, 2019/04. Gavin N. Petrie, Kiri L. Wills, Fabiana Piscitelli, Reem Smoum, Cheryl L. Limebeer, Erin M. Rock, Ashlyn E. Humphrey, Madeleine Sheppard-Perkins, Aron H. Lichtman, Raphael Mechoulam, Vincenzo Di Marzo, Linda A. Parker. DOI 10.1007/s00213-019-05237-9
Identification and characterization of phytocannabinoids as novel dual PPARα/γ agonists by a computational and in vitro experimental approach Biochimica et Biophysica Acta (BBA) - General Subjects, 2019/03. Enrico D'Aniello, Tariq Fellous, Fabio Arturo Iannotti, Alessandra Gentile, Marco Allarà, Francesca Balestrieri, Roy Gray, Pietro Amodeo, Rosa Maria Vitale, Vincenzo Di Marzo. DOI 10.1016/j.bbagen.2019.01.002
Peripubertal cannabidiol treatment rescues behavioral and neurochemical abnormalities in the MAM model of schizophrenia Neuropharmacology, 2019/03. Tibor Stark, Jana Ruda-Kucerova, Fabio Arturo Iannotti, Claudio D'Addario, Roberta Di Marco, Vladimir Pekarik, Eva Drazanova, Fabiana Piscitelli, Monica Bari, Zuzana Babinska, Giovanni Giurdanella, Martina Di Bartolomeo, Salvatore Salomone, Alexandra Sulcova, Mauro Maccarrone, Carsten T. Wotjak, Zenon Starcuk, Filippo Drago, Raphael Mechoulam, Vincenzo Di Marzo, Vincenzo Micale. DOI 10.1016/j.neuropharm.2018.11.035
Synthesis of novel 2-(1-adamantanylcarboxamido)thiophene derivatives. Selective cannabinoid type 2 (CB2) receptor agonists as potential agents for the treatment of skin inflammatory disease European Journal of Medicinal Chemistry, 2019/01. Claudia Mugnaini, Alessandro Rabbito, Antonella Brizzi, Nastasja Palombi, Stefania Petrosino, Roberta Verde, Vincenzo Di Marzo, Alessia Ligresti, Federico Corelli. DOI 10.1016/j.ejmech.2018.09.070
In Silico Identification and Experimental Validation of (−)-Muqubilin A, a Marine Norterpene Peroxide, as PPARα/γ-RXRα Agonist and RARα Positive Allosteric Modulator Marine Drugs, 2019/02. Enrico D’Aniello, Fabio Arturo Iannotti, Lauren G. Falkenberg, Andrea Martella, Alessandra Gentile, Fabrizia De Maio, Maria Letizia Ciavatta, Margherita Gavagnin, Joshua Waxman, Vincenzo Di Marzo, Pietro Amodeo, ROSA MARIA VITALE. DOI 10.3390/md17020110
Effects of diisononyl phthalate (DiNP) on the endocannabinoid and reproductive systems of male gilthead sea bream (Sparus aurata) during the spawning season Archives of Toxicology, 2019/01/02. Isabel Forner-Piquer, Constantinos C. Mylonas, Ioannis Fakriadis, Maria Papadaki, Fabiana Piscitelli, Vincenzo Di Marzo, Josep Calduch-Giner, Jaume Pérez-Sánchez, Oliana Carnevali. DOI 10.1007/s00204-018-2378-6
Intestinal epithelial N-acylphosphatidylethanolamine phospholipase D links dietary fat to metabolic adaptations in obesity and steatosis Nature Communications, 2019/01. Amandine Everard, Hubert Plovier, Marialetizia Rastelli, Matthias Van Hul, Alice de Wouters d’Oplinter, Lucie Geurts, Céline Druart, Sylvie Robine, Nathalie M. Delzenne, Giulio G. Muccioli, Willem M. de Vos, Serge Luquet, Nicolas Flamand, Vincenzo Di Marzo, Patrice D. Cani. DOI 10.1038/s41467-018-08051-7
Summary of the International Conference on Onco-Nephrology: an emerging field in medicine Kidney International, 2019. Capasso, A., Benigni, A., Capitanio, U., Danesh, F.R., Di Marzo, V., Gesualdo, L., Grandaliano, G., Jaimes, E.A., Malyszko, J., Perazella, M.A., Qian, Q., Ronco, P., Rosner, M.H., Trepiccione, F., Viggiano, D., Zoccali, C., Capasso, G., Akitaka, A., Alahoti, A., Alexander, T.R., Altucci, L., Amer, H., Barone, V., Eri, K., Biancone, L., Bonventre, J.V., Camussi, G., Ciardiello, F., Caraglia, M., Cartenì, G., Cervantes, A., Citterio, F., Cosmai, L., Daniele, B., D'Errico, A., De Vita, F., Ereditato, A., Falco, G., Fouque, D., Franco, R., Gallieni, M., Gambaro, G., Kuo, C., Launay-Vacher, V., Maiello, E., Mallamaci, F., Malysxko, J., Marino, G., Martinelli, E., Matarese, G., Matsubara, T., Messa, P., Messina, C., Mirone, V., Morgillo, F., Costa, A.N., Orditura, M., Pani, A., Perazella, M.A., Perna, A., Pisano, C., Pitts, T., Porta, C., Procopio, G., Remuzzi, G., Russo, D., Siu, L.L., Stadler, W., Troiani, T., Weisz, A., Więcek, A., Xiaoqiang, D., Zecchino, O.. DOI 10.1016/j.kint.2019.04.043
Ultra-micronized palmitoylethanolamide rescues the cognitive decline-associated loss of neural plasticity in the neuropathic mouse entorhinal cortex-dentate gyrus pathway Neurobiology of Disease, 2019/01. Serena Boccella, Claudia Cristiano, Rosaria Romano, Monica Iannotta, Carmela Belardo, Antonio Farina, Francesca Guida, Fabiana Piscitelli, Enza Palazzo, Mariacristina Mazzitelli, Roberta Imperatore, Lea Tunisi, Vito de Novellis, Luigia Cristino, Vincenzo Di Marzo, Antonio Calignano, Sabatino Maione, Livio Luongo. DOI 10.1016/j.nbd.2018.09.023
Palmitoylethanolamide counteracts substance P-induced mast cell activation in vitro by stimulating diacylglycerol lipase activity Journal of Neuroinflammation, 2019. Petrosino, S., Schiano Moriello, A., Verde, R., Allarà, M., Imperatore, R., Ligresti, A., Mahmoud, A.M., Peritore, A.F., Iannotti, F.A., Di Marzo, V.. DOI 10.1186/s12974-019-1671-5
Rapid and concomitant gut microbiota and endocannabinoidome response to diet-induced obesity in mice mSystems, 2019. Lacroix, S., Pechereau, F., Leblanc, N., Boubertakh, B., Houde, A., Martin, C., Flamand, N., Silvestri, C., Raymond, F., Marzo, V.D., Veilleuxa, A.. DOI 10.1128/mSystems.00407-19
5th EFLM-UEMS European Joint Congress in Laboratory Medicine Clinical Chemistry and Laboratory Medicine (CCLM), 2018/10. DOI 10.1515/cclm-2018-1038
The Expanded Endocannabinoid System/Endocannabinoidome as a Potential Target for Treating Diabetes Mellitus Current Diabetes Reports, 2019. Veilleux, A., Di Marzo, V., Silvestri, C.. DOI 10.1007/s11892-019-1248-9
Reversal of albuminuria by combined AM6545 and perindopril therapy in experimental diabetic nephropathy British Journal of Pharmacology, 2018/12/06. F Barutta, S Bellini, R Mastrocola, R Gambino, F Piscitelli, V di Marzo, B Corbetta, VK Vemuri, A Makriyannis, L Annaratone, G Bruno, G Gruden. DOI 10.1111/bph.14495
Fishing for Targets of Alien Metabolites: A Novel Peroxisome Proliferator-Activated Receptor (PPAR) Agonist from a Marine Pest Marine Drugs, 2018/11. Rosa Maria Vitale, Enrico D'Aniello, Stefania Gorbi, Andrea Martella, Cristoforo Silvestri, Maria Elisa Giuliani, Tariq Fellous, Alessandra Gentile, Marianna Carbone, Adele Cutignano, Laura Grauso, Laura Magliozzi, Gianluca Polese, BIAGIO D'ANIELLO, Fanny Defranoux, Serena Felline, Antonio Terlizzi, Antonio Calignano, Francesco Regoli, Vincenzo Di Marzo, Pietro Amodeo, Ernesto Mollo. DOI 10.3390/md16110431
Elongation of the Hydrophobic Chain as a Molecular Switch: Discovery of Capsaicin Derivatives and Endogenous Lipids as Potent Transient Receptor Potential Vanilloid Channel 2 Antagonists Journal of Medicinal Chemistry, 2018/09/27. Aniello Schiano Moriello, Silvia López Chinarro, Olalla Novo Fernández, Jordi Eras, Pietro Amodeo, Ramon Canela-Garayoa, Rosa Maria Vitale, Vincenzo Di Marzo, Luciano De Petrocellis. DOI 10.1021/acs.jmedchem.8b00734
Disruption of the gonadal endocannabinoid system in zebrafish exposed to diisononyl phthalate Environmental Pollution, 2018/10. Isabel Forner-Piquer, Stefania Santangeli, Francesca Maradonna, Alessandro Rabbito, Fabiana Piscitelli, Hamid R. Habibi, Vincenzo Di Marzo, Oliana Carnevali. DOI 10.1016/j.envpol.2018.05.007
Endocrine disruptors in the diet of male Sparus aurata: Modulation of the endocannabinoid system at the hepatic and central level by Di-isononyl phthalate and Bisphenol A Environment International, 2018/10. Isabel Forner-Piquer, Constantinos C. Mylonas, Josep Calduch-Giner, Francesca Maradonna, Giorgia Gioacchini, Marco Allarà, Fabiana Piscitelli, Vincenzo Di Marzo, Jaume Pérez-Sánchez, Oliana Carnevali. DOI 10.1016/j.envint.2018.06.011
Δ9-tetrahydrocannabivarin impairs epithelial calcium transport through inhibition of TRPV5 and TRPV6 Pharmacological Research, 2018/10. Annelies Janssens, Cristoforo Silvestri, Andrea Martella, Jo M. Vanoevelen, Vincenzo Di Marzo, Thomas Voets. DOI 10.1016/j.phrs.2018.08.021
Genetic and pharmacological regulation of the endocannabinoid CB1 receptor in Duchenne muscular dystrophy Nature Communications, 2018/09. Fabio A. Iannotti, Ester Pagano, Ombretta Guardiola, Simone Adinolfi, Valentina Saccone, Silvia Consalvi, Fabiana Piscitelli, Elisabetta Gazzerro, Giuseppe Busetto, Diego Carrella, Raffaele Capasso, Pier Lorenzo Puri, Gabriella Minchiotti, Vincenzo Di Marzo. DOI 10.1038/s41467-018-06267-1
Effects of non-euphoric plant cannabinoids on muscle quality and performance of dystrophic mdx mice British Journal of Pharmacology, 2018/09/09. Fabio Arturo Iannotti, Ester Pagano, Aniello Schiano Moriello, Filomena Grazia Alvino, Nicolina Cristina Sorrentino, Luca D'Orsi, Elisabetta Gazzerro, Raffaele Capasso, Elvira De Leonibus, Luciano De Petrocellis, Vincenzo Di Marzo. DOI 10.1111/bph.14460
Author Correction: CB1 receptor activation induces intracellular Ca2+ mobilization and 2-arachidonoylglycerol release in rodent spinal cord astrocytes Scientific Reports, 2018/09/07. Zoltán Hegyi, Tamás Oláh, Áron Kőszeghy, Fabiana Piscitelli, Krisztina Holló, Balázs Pál, László Csernoch, Vincenzo Di Marzo, Miklós Antal. DOI 10.1038/s41598-018-30573-9
FAAH-Catalyzed C–C Bond Cleavage of a New Multitarget Analgesic Drug ACS Chemical Neuroscience, 2018/09. Alessia Ligresti, Cristoforo Silvestri, Rosa Maria Vitale, Jose L. Martos, Fabiana Piscitelli, Jenny W. Wang, Marco Allarà, Robert W. Carling, Livio Luongo, Francesca Guida, Anna Illiano, Angela Amoresano, Sabatino Maione, Pietro Amodeo, David F. Woodward, Vincenzo Di Marzo, Gennaro Marino. DOI 10.1021/acschemneuro.8b00315
New approaches and challenges to targeting the endocannabinoid system Nature Reviews Drug Discovery, 2018/08. Vincenzo Di Marzo. DOI 10.1038/nrd.2018.115
Development of Potent Inhibitors of Fatty Acid Amide Hydrolase Useful for the Treatment of Neuropathic Pain ChemMedChem, 2018/08. Margherita Brindisi, Giuseppe Borrelli, Simone Brogi, Alessandro Grillo, Samuele Maramai, Marco Paolino, Mascia Benedusi, Alessandra Pecorelli, Giuseppe Valacchi, Lorenzo Di Cesare Mannelli, Carla Ghelardini, Marco Allarà, Alessia Ligresti, Patrizia Minetti, Giuseppe Campiani, Vincenzo di Marzo, Stefania Butini, Sandra Gemma. DOI 10.1002/cmdc.201800397
Endocannabinoid Tone Regulates Human Sebocyte Biology Journal of Investigative Dermatology, 2018/08. Nóra Zákány, Attila Oláh, Arnold Markovics, Erika Takács, Andrea Aranyász, Simon Nicolussi, Fabiana Piscitelli, Marco Allarà, Ágnes Pór, Ilona Kovács, Christos C. Zouboulis, Jürg Gertsch, Vincenzo Di Marzo, Tamás Bíró, Tamás Szabó. DOI 10.1016/j.jid.2018.02.022
Experimental ischemia/reperfusion model impairs endocannabinoid signaling and Na+/K+ ATPase expression and activity in kidney proximal tubule cells Biochemical Pharmacology, 2018/08. Luzia S. Sampaio, Fabio A. Iannotti, Luciana Veneziani, Rosa T. Borelli-Tôrres, Fabrizia De Maio, Fabiana Piscitelli, Ricardo A.M. Reis, Vincenzo Di Marzo, Marcelo Einicker-Lamas. DOI 10.1016/j.bcp.2018.06.005
The Involvement of the Endocannabinoid System in the Peripheral Antinociceptive Action of Ketamine The Journal of Pain, 2018/05. Renata C.M. Ferreira, Marina G.M. Castor, Fabiana Piscitelli, Vincenzo Di Marzo, Igor D.G. Duarte, Thiago R.L. Romero. DOI 10.1016/j.jpain.2017.12.002
Role of Bisphenol A on the Endocannabinoid System at central and peripheral levels: Effects on adult female zebrafish Chemosphere, 2018/08. Isabel Forner-Piquer, Stefania Santangeli, Francesca Maradonna, Roberta Verde, Fabiana Piscitelli, Vincenzo di Marzo, Hamid R. Habibi, Oliana Carnevali. DOI 10.1016/j.chemosphere.2018.04.078
CB1 receptor activation induces intracellular Ca2+ mobilization and 2-arachidonoylglycerol release in rodent spinal cord astrocytes Scientific Reports, 2018/07. Zoltán Hegyi, Tamás Oláh, Áron Kőszeghy, Fabiana Piscitelli, Krisztina Holló, Balázs Pál, László Csernoch, Vincenzo Di Marzo, Miklós Antal. DOI 10.1038/s41598-018-28763-6
Overlapping Distribution of Orexin and Endocannabinoid Receptors and Their Functional Interaction in the Brain of Adult Zebrafish Frontiers in Neuroanatomy, 2018/07. Roberta Imperatore, Livia D’Angelo, Omid Safari, Hamidreza Ahmadniaye Motlagh, Fabiana Piscitelli, Paolo de Girolamo, Luigia Cristino, Ettore Varricchio, Vincenzo di Marzo, Marina Paolucci. DOI 10.3389/fnana.2018.00062
Effects of repeated long-term psychosocial stress and acute cannabinoid exposure on mouse corticostriatal circuitries: Implications for neuropsychiatric disorders CNS Neuroscience & Therapeutics, 2018/01. Jordi Tomas-Roig, Fabiana Piscitelli, Vanesa Gil, Ester Quintana, Lluís l. Ramió-Torrentà, Jose Antonio del Río, Timothy Patrick Moore, Hope Agbemenyah, Gabriela Salinas, Claudia Pommerenke, Stephan Lorenzen, Tim Beißbarth, Sigrid Hoyer-Fender, Vincenzo Di Marzo, Ursula Havemann-Reinecke. DOI 10.1111/cns.12810
Anti-inflammatory Properties of Cannabidiol, a Nonpsychotropic Cannabinoid, in Experimental Allergic Contact Dermatitis Journal of Pharmacology and Experimental Therapeutics, 2018/04/09. Stefania Petrosino, Roberta Verde, Massimo Vaia, Marco Allarà, Teresa Iuvone, Vincenzo Di Marzo. DOI 10.1124/jpet.117.244368
Oral Ultramicronized Palmitoylethanolamide: Plasma and Tissue Levels and Spinal Anti-hyperalgesic Effect Frontiers in Pharmacology, 2018/03. Stefania Petrosino, Marika Cordaro, Roberta Verde, Aniello Schiano Moriello, Gabriele Marcolongo, Carlo Schievano, Rosalba Siracusa, Fabiana Piscitelli, Alessio F. Peritore, Rosalia Crupi, Daniela Impellizzeri, Emanuela Esposito, Salvatore Cuzzocrea, Vincenzo Di Marzo. DOI 10.3389/fphar.2018.00249
Antibiotic-induced microbiota perturbation causes gut endocannabinoidome changes, hippocampal neuroglial reorganization and depression in mice Brain, Behavior, and Immunity, 2018/01. F. Guida, F. Turco, M. Iannotta, D. De Gregorio, I. Palumbo, G. Sarnelli, A. Furiano, F. Napolitano, S. Boccella, L. Luongo, M. Mazzitelli, A. Usiello, F. De Filippis, F.A. Iannotti, F. Piscitelli, D. Ercolini, V. de Novellis, V. Di Marzo, R. Cuomo, S. Maione. DOI 10.1016/j.bbi.2017.09.001
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